发明名称 FUSED HETEROCYCLIC COMPOUNDS AS OREXIN RECEPTOR MODULATORS
摘要 Certain disubstituted 3,8-diaza-bicyclo[4.2.0]octane and 3,6-diazabicyclo [3.2.0]heptane are described, which are useful as orexin inhibitors. Such compounds may be useful in pharmaceutical compositions and methods for the treatment of diseased states, disorders, and conditions mediated by orexin activity, such as insomnia.
申请公布号 WO2011050202(A1) 申请公布日期 2011.04.28
申请号 WO2010US53611 申请日期 2010.10.21
申请人 JANSSEN PHARMACEUTICA NV;BRANSTETTER, BRYAN, JAMES;LETAVIC, MICHAEL, A.;LY, KIEV, S.;RUDOLPH, DALE, A.;SAVALL, BRAD, M.;SHAH, CHANDRAVADAN, R.;SHIREMAN, BROCK, T. 发明人 BRANSTETTER, BRYAN, JAMES;LETAVIC, MICHAEL, A.;LY, KIEV, S.;RUDOLPH, DALE, A.;SAVALL, BRAD, M.;SHAH, CHANDRAVADAN, R.;SHIREMAN, BROCK, T.
分类号 C07D471/04;A61K31/4353;A61P25/00;C07D487/04 主分类号 C07D471/04
代理机构 代理人
主权项
地址