发明名称 PYRAZOLOTHIAZOLE COMPOUND
摘要 <p>A compound represented by formula (I) or a pharmacologically acceptable salt thereof, which has an excellent antagonistic activity on a CRF receptor. [In the formula, X represents a nitrogen atom or CH; R1 represents -A11-A12; A11 represents a single bond or an alkylene group; A12 represents a hydrogen atom, an alkyl group or a cycloalkyl group; R2 represents -A21-A22; A21 represents a single bond or an alkylene group; A22 represents a hydrogen atom, an alkyl group, a cycloalkyl group, a non-aromatic heterocyclic group, a heteroaryl group or the like; R3 represents an alkyl group, a cycloalkyl group, an alkoxy group, a cycloalkoxyalkyl group, a dialkylamino group, a halogen atom, a cyano group, a formyl group, a carboxyl group or the like; R4 represents a hydrogen atom or an alkoxy group; R5 represents a halogen atom, an alkyl group or an alkoxy group; R6 represents a hydrogen atom, an alkyl group, an alkoxy group, an alkylthio group, an alkylsulfinyl group or the like; and R7 represents an alkyl group, an alkoxy group or an alkylthio group.]</p>
申请公布号 WO2011043381(A1) 申请公布日期 2011.04.14
申请号 WO2010JP67556 申请日期 2010.10.06
申请人 EISAI R&D MANAGEMENT CO., LTD.;SHIN KOGYOKU;TERAUCHI TARO;TAKAHASHI YOSHINORI;HASHIZUME MINAKO;TAKEDA KUNITOSHI;SHIKATA KODO;INOMATA AKIRA 发明人 SHIN KOGYOKU;TERAUCHI TARO;TAKAHASHI YOSHINORI;HASHIZUME MINAKO;TAKEDA KUNITOSHI;SHIKATA KODO;INOMATA AKIRA
分类号 C07D513/04;A61K31/429;A61K31/4439;A61P1/00;A61P1/04;A61P9/10;A61P9/12;A61P25/08;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P43/00 主分类号 C07D513/04
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