发明名称 Amorphous object of cinnamide compound
摘要 An amorphous object of (3E)-1-[l(s)-1-(4-fluorophenyl)ethyl]-3-[3-methoxy-4-(4methyl-1H-imidazol-1-yl)benzylidene]piperidine-2-one, which is represented by the formula (1) and has A&bgr;-production inhibitory activity. The amorphous object has such satisfactory properties that it has excellent solubility, is stable, does not readily become a crystalline form, and has low hygroscopicity. It is hence suitable for use in pharmaceutical preparations.
申请公布号 US7923563(B2) 申请公布日期 2011.04.12
申请号 US20050663550 申请日期 2005.10.25
申请人 EISAI R&D MANAGEMENT CO., LTD. 发明人 KUSHIDA IKUO;DOI ERIKO;ITO KOICHI
分类号 C07D401/06 主分类号 C07D401/06
代理机构 代理人
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