发明名称 METHOD FOR PURIFYING 4-AMINO-5-CHLORO-2-ETHOXY-N-[[4-(4-FLUOROBENZYL)-2-MORPHOLINYL]METHYL]BENZAMIDE
摘要 PROBLEM TO BE SOLVED: To provide a method for preparing 4-amino-5-chloro-2-ethoxy-N-[[4-(4-fluorobenzyl)-2-morpholinyl]methyl]benzamide in high yield with high purity. SOLUTION: The method includes steps of dissolving a crude matter containing 4-amino-5-chloro-2-ethoxy-N-[[4-(4-fluorobenzyl)-2-morpholinyl]methyl]benzamide in a solvent containing an amide solvent and subsequently crystallizing 4-amino-5-chloro-2-ethoxy-N-[[4-(4-fluorobenzyl)-2-morpholinyl]methyl]benzamide from the resulting solution. COPYRIGHT: (C)2011,JPO&INPIT
申请公布号 JP2011068611(A) 申请公布日期 2011.04.07
申请号 JP20090222051 申请日期 2009.09.28
申请人 TOKUYAMA CORP 发明人 KAMIZONO HIROYUKI;MIYAOKU TAKAYUKI;TANAKA KENJI
分类号 C07D265/30 主分类号 C07D265/30
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