发明名称 |
GAIN-OF-FUNCTION BCL-2 INHIBITORS |
摘要 |
Compounds are described that are useful for treating an apoptosis-associated disease, which are specifically cytotoxic to tumor cells that are overexpressing BcI-XL, and are much less cytotoxic in isogenic cells that are not overexpressing BcI-XL. Methods of using such compounds to treat apoptosis-associated disease is also described. |
申请公布号 |
WO2011041737(A2) |
申请公布日期 |
2011.04.07 |
申请号 |
WO2010US51208 |
申请日期 |
2010.10.01 |
申请人 |
FRED HUTCHINSON CANCER RESEARCH CENTER;HOCKENBERY, DAVID;SIMON, JULIAN |
发明人 |
HOCKENBERY, DAVID;SIMON, JULIAN |
分类号 |
C07D213/53;A61K31/15;C07C251/80;C07D213/77 |
主分类号 |
C07D213/53 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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