<p>The invention discloses 1-N-substituted-6-(hetero)aryl-1H-thieno[3,2-d]pyrimidin-4-one derivatives of formula (I) wherein R1, R2, R3 and R4 are as defined herein that inhibit Hepatitis C virus NS5b polymerase inhibitors. Also disclosed are compositions and methods for treating an HCV infection and inhibiting HCV replication.</p>
申请公布号
WO2011036128(A1)
申请公布日期
2011.03.31
申请号
WO2010EP63832
申请日期
2010.09.21
申请人
F. HOFFMANN-LA ROCHE AG;BROKA, CHRIS ALLEN;HENDRICKS, ROBERT THAN;MAAG, HANS;SMITH, DAVID BERNARD;WANNER, JUTTA
发明人
BROKA, CHRIS ALLEN;HENDRICKS, ROBERT THAN;MAAG, HANS;SMITH, DAVID BERNARD;WANNER, JUTTA