发明名称 PROCESSES FOR PREPARING TETRAHYDROISOQUINOLINES
摘要 Disclosed are processes for preparing tetrahydroisoquinolines, intermediates useful in the preparation of tetrahydroisoquinolines, processes for preparing such intermediates, and a crystalline form of 6-[(4S)-2-methyl-4-(naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine. Also disclosed are pharmaceutical compositions comprising tetrahydroisoquinolines, methods of using tetrahydroisoquinolines in the treatment of depression and other conditions and methods for obtaining the crystalline form.
申请公布号 US2011077400(A1) 申请公布日期 2011.03.31
申请号 US20090995776 申请日期 2009.06.04
申请人 BRISTOL-MYERS SQUIBB COMPANY AND ALBANY MOLECULARRESEARCH, INC 发明人 LOBBEN PAUL;ZHAO RULIN;WANG BEI;CHEN BANG-CHI;LIU SHUANG;HU MIN;YANG YUH-LIN ALLEN;ISHERWOOD MATTHEW;AMIN RASIDUL;CUI WENGE
分类号 C07D403/10;C07C211/26;C07D217/02;C07D237/02;C07F5/02 主分类号 C07D403/10
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