发明名称 |
METHODS FOR ISOLATING PROPARGYLATED AMINOINDANS |
摘要 |
A process for isolating from a reaction mixture a salt of a mono-propargylated aminoindan, a process for isolating from a reaction mixture a crystalline diastereomeric salt of a mono-propargylated aminoindan, and a process for isolating from a reaction mixture a salt of enantiomerically pure N-propargyl-1-aminoindan or a salt of enantiomerically pure 6-(N-methyl, N-ethyl-carbamoyloxy)-N'-propargyl-1-aminoindan. The corresponding products are also disclosed. |
申请公布号 |
EP1954667(A4) |
申请公布日期 |
2011.03.23 |
申请号 |
EP20060837655 |
申请日期 |
2006.11.15 |
申请人 |
TEVA PHARMACEUTICAL INDUSTRIES LTD |
发明人 |
FRENKEL, ANTON;LIDOR-HADAS, RAMY;GUREVICH, EDUARD;ATTILI, GSAN |
分类号 |
C07C209/84 |
主分类号 |
C07C209/84 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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