发明名称 |
Organic compound and method for producing radioactive halogen-labeled organic compound using the same |
摘要 |
It is intended to provide a labeling precursor compound used for selectively producing radioactive halogen-substituted syn-1-amino-3-cyclobutane-carboxylic acids, and to provide a process for producing a radioactive halogen-substituted syn-1-amino-3-cyclobutane-carboxylic acid using the labeling precursor compound. A labeling precursor is used in which a phthalimide group is used as a protective group for protecting the amino group. The syn-form of the radioactive halogen-substituted 1-amino-3-cyclobutane-carboxylic acid can be selectively produced by labeling the labeling precursor with a radioactive halogen followed by deprotecting.
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申请公布号 |
US7910745(B2) |
申请公布日期 |
2011.03.22 |
申请号 |
US20060915267 |
申请日期 |
2006.05.15 |
申请人 |
NIHON MEDI-PHYSICS CO., LTD. |
发明人 |
TOYAMA MASAHITO;KUROSAKI FUMIE;HAYASHI AKIO;ITO OSAMU |
分类号 |
C07D285/01;C07C61/04;C07D207/404;C07D209/48 |
主分类号 |
C07D285/01 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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