发明名称 4- (PYRIMIDIN-2-YL) -PIPERAZINE AND 4- (PYRIMIDIN-2-YL) -PIPERIDINE DERIVATIVES AS GPR119 MODULATORS
摘要 <p>A compound of formula (I) or a pharmaceutically acceptable salt thereof, processes for preparing such compounds, their use as GPR119 modulators, methods for their therapeutic use, particularly in the treatment of obesity and diabetes mellitus, and pharmaceutical compositions containing them.</p>
申请公布号 WO2011030139(A1) 申请公布日期 2011.03.17
申请号 WO2010GB51483 申请日期 2010.09.07
申请人 ASTRAZENECA AB;ASTRAZENECA UK LIMITED;BIRCH, ALAN, MARTIN;BROO, DAN, ANDERS;BUTLIN, ROGER, JOHN;CLARKE, DAVID, STEPHEN;DAVIDSSON, OJVIND, PERCY;DE LA MOTTE, HANNA;JOHANSSON, KJELL, ERIK;LEACH, ANDREW;MACFAUL, PHILIP, ALEXANDER;O'DONNELL, CHARLES, JOHN;SCOTT, JAMES, STEWART;WHITTAMORE, PAUL, ROBERT, OWEN 发明人 BIRCH, ALAN, MARTIN;BROO, DAN, ANDERS;BUTLIN, ROGER, JOHN;CLARKE, DAVID, STEPHEN;DAVIDSSON, OJVIND, PERCY;DE LA MOTTE, HANNA;JOHANSSON, KJELL, ERIK;LEACH, ANDREW;MACFAUL, PHILIP, ALEXANDER;O'DONNELL, CHARLES, JOHN;SCOTT, JAMES, STEWART;WHITTAMORE, PAUL, ROBERT, OWEN
分类号 C07D239/47;A61K31/506;A61P3/04;A61P3/10;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D403/14;C07D413/12;C07D413/14 主分类号 C07D239/47
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