发明名称 PREPARATION OF RALOXIFENE AND ITS SALTS
摘要 The invention provides processes for the preparation of pure raloxifene or its salts, involving hydrolyzing 6-methylsulfonyloxy-2-[(4-methylsulfonyloxy)-phenyl]-3-[4(2-(piperidinyl)ethoxy)benzoyl]benzothiophene hydrochloride, using an aqueous base.
申请公布号 WO2011029088(A2) 申请公布日期 2011.03.10
申请号 WO2010US47966 申请日期 2010.09.07
申请人 DR. REDDY'S LABORATORIES LTD.;DR. REDDY'S LABORATORIES, INC.;SANDEEP, MOHANTY;GADDAMEEDHI, PRASHANTH REDDY;MOHAN, GUNTI MURALI;REDDY, KESAVA;BATHINI, PAVAN KUMAR;KOMMAREDDY, VENKATESWARA REDDY 发明人 SANDEEP, MOHANTY;GADDAMEEDHI, PRASHANTH REDDY;MOHAN, GUNTI MURALI;REDDY, KESAVA;BATHINI, PAVAN KUMAR;KOMMAREDDY, VENKATESWARA REDDY
分类号 C07D409/12;A61K31/4535;A61P5/32 主分类号 C07D409/12
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