发明名称 COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS
摘要 The invention relates to compounds of structural formula (I): or a pharmaceutically acceptable salt, solvate, clathrate, and prodrug thereof, wherein Ra, Rb, and R2 are defined herein. These compounds inhibit tubulin polymerization and/or target vasculature and are useful for treating proliferative disorders, such as cancer.
申请公布号 US2011059893(A1) 申请公布日期 2011.03.10
申请号 US20100883883 申请日期 2010.09.16
申请人 SYNTA PHARMACEUTICALS CORP. 发明人 SUN LIJUN;BORELLA CHRISTOPHER;LI HAO;JIANG JUN;CHEN SHOUJUN;KOYA KEIZO;INOUE TAKAYO;DU ZHENJIAN;FOLEY KEVIN;WU YAMING;ZHANG MEI;YING WEIWEN
分类号 A61K38/06;A61K31/42;A61K31/422;A61K31/4439;A61K31/4709;A61K31/4725;A61K31/501;A61K31/675;A61P7/00;A61P27/02;A61P35/00;C07D261/08;C07D413/04;C07D413/10;C07F9/09;C07K5/08 主分类号 A61K38/06
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