发明名称 |
CRYSTALLINE MONOHYDRATE, METHOD FOR PRODUCING THE SAME AND THE USE THEREOF IN THE PRODUCTION OF A MEDICAMENT |
摘要 |
Crystalline monohydrate (I) of tiotropium bromide ((1alpha ,2beta ,4beta ,5alpha ,7beta )-7-(2-hydroxy-2,2-di(2-thienyl)acetoxy)-9,9-dimethyl-3-oxa-9-azonia-tricyclo[3.3.1.0 2>.4]nonane bromide) is new. An independent claim is also included for the preparation of (I). ACTIVITY : Antiinflammatory; antiasthmatic. MECHANISM OF ACTION : Anticholinergic. |
申请公布号 |
PL207870(B1) |
申请公布日期 |
2011.02.28 |
申请号 |
PL20010366041 |
申请日期 |
2001.09.28 |
申请人 |
BOEHRINGER INGELHEIM PHARMA GMBH & CO.KG |
发明人 |
BANHOLZER ROLF;SIEGER PETER;KULINNA CHRISTIAN;TRUNK MICHAEL;GRAULICH MANFRED LUDWIG AUGUST;SPECHT PETER;MEISSNER HELMUT;MATHES ANDREAS |
分类号 |
C07D451/10;A61K9/14;A61K9/72;A61K31/439;A61K31/46;A61P11/00;A61P11/06;A61P43/00;C07D451/14 |
主分类号 |
C07D451/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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