发明名称 |
PROCESS FOR PRODUCING BENZO[B][1,4]DIAZEPINE-2,4-DIONE COMPOUND |
摘要 |
<p>Provided is a process for industrially advantageously, easily, and efficiently producing a key intermediate for a benzo[b][1,4]diazepine-2,4-dione compound that is a therapeutic agent for arrhythmia. The process is for producing a compound represented by general formula (1) (wherein R1, R2, R3, and R4 are the same or different and each represents a hydrogen atom or a lower alkyl), and is characterized by eliminating the protective group (R5) of a compound represented by general formula (2) (wherein R1, R2, R3, and R4 are the same as defined above, and R5 represents a protective group for the hydroxy group).</p> |
申请公布号 |
WO2011021676(A1) |
申请公布日期 |
2011.02.24 |
申请号 |
WO2010JP64040 |
申请日期 |
2010.08.20 |
申请人 |
OTSUKA PHARMACEUTICAL CO., LTD.;TSUJIMORI, HISAYUKI;TAIRA, SHINICHI;YUKAWA, HIROTAKA;ABE, KAORU |
发明人 |
TSUJIMORI, HISAYUKI;TAIRA, SHINICHI;YUKAWA, HIROTAKA;ABE, KAORU |
分类号 |
C07D243/12 |
主分类号 |
C07D243/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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