发明名称 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
摘要 <p>Compounds of Formula I wherein R1, R2, X, and Y are as defined herein, or a tautomer, optical isomer, prodrug, co-crystal, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.</p>
申请公布号 WO2009149139(A8) 申请公布日期 2011.02.24
申请号 WO2009US46058 申请日期 2009.06.03
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG;BETAGERI, RAJASHEKHAR;BOSANAC, TODD;BURKE, MICHAEL, JASON;HARCKEN, CHRISTIAN;KIM, SOOJIN;KUZMICH, DANIEL;LEE, THOMAS, WAI-HO;LI, ZHIBIN;LIU, PINGRONG;LORD, JOHN;RAZAVI, HOSSEIN;REEVES, JONATHAN, TIMOTHY;THOMSON, DAVID 发明人 BETAGERI, RAJASHEKHAR;BOSANAC, TODD;BURKE, MICHAEL, JASON;HARCKEN, CHRISTIAN;KIM, SOOJIN;KUZMICH, DANIEL;LEE, THOMAS, WAI-HO;LI, ZHIBIN;LIU, PINGRONG;LORD, JOHN;RAZAVI, HOSSEIN;REEVES, JONATHAN, TIMOTHY;THOMSON, DAVID
分类号 C07D471/04;A61K31/437;A61P5/44;A61P5/46 主分类号 C07D471/04
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