发明名称 |
REAGENT AND METHOD FOR PREPARING LPS ANTAGONIST B1287 AND STEREOISOMER THEREOF |
摘要 |
PROBLEM TO BE SOLVED: To provide methods for preparing LPS (linear programming system) antagonist lipodisaccharide B1287 and stereoisomers thereof. SOLUTION: The invention provides methods for preparing LPS antagonist lipodisaccharide B1287 useful in the prophylactic and affirmative treatment of endotoxemia shown by formula, and stereoisomers thereof. Also there are provided useful synthetic intermediates. COPYRIGHT: (C)2011,JPO&INPIT
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申请公布号 |
JP2011037885(A) |
申请公布日期 |
2011.02.24 |
申请号 |
JP20100230114 |
申请日期 |
2010.10.12 |
申请人 |
EISAI R & D MANAGEMENT CO LTD |
发明人 |
FAN RULIN |
分类号 |
C07H1/02;A61K31/7024;A61P7/00;A61P31/04;C07H3/04;C07H9/04;C07H15/04;C07H15/12 |
主分类号 |
C07H1/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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