发明名称 REAGENT AND METHOD FOR PREPARING LPS ANTAGONIST B1287 AND STEREOISOMER THEREOF
摘要 PROBLEM TO BE SOLVED: To provide methods for preparing LPS (linear programming system) antagonist lipodisaccharide B1287 and stereoisomers thereof. SOLUTION: The invention provides methods for preparing LPS antagonist lipodisaccharide B1287 useful in the prophylactic and affirmative treatment of endotoxemia shown by formula, and stereoisomers thereof. Also there are provided useful synthetic intermediates. COPYRIGHT: (C)2011,JPO&INPIT
申请公布号 JP2011037885(A) 申请公布日期 2011.02.24
申请号 JP20100230114 申请日期 2010.10.12
申请人 EISAI R & D MANAGEMENT CO LTD 发明人 FAN RULIN
分类号 C07H1/02;A61K31/7024;A61P7/00;A61P31/04;C07H3/04;C07H9/04;C07H15/04;C07H15/12 主分类号 C07H1/02
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