发明名称 1,2,4-Triazolylaminoaryl (heteroaryl) sulfonamide derivatives
摘要 1,2,4-Triazolylaminoaryl(heteroaryl)sulfonamide derivatives of formula (I), pharmaceutically acceptable salts thereof, processes for the manufacture of 1,2,4-triazolylaminoaryl(heteroaryl)sulfonamide derivatives and pharmaceutical compositions containing 1,2,4-triazolylaminoaryl(heteroaryl)sulfonamide derivatives are disclosed: The 1,2,4-triazolylaminoaryl(heteroaryl)sulfonamide derivatives of formula (I) possess cell cycle inhibitory activity and are accordingly useful for their anti cell proliferation (such as anti cancer) activity.
申请公布号 US7888380(B2) 申请公布日期 2011.02.15
申请号 US20050245314 申请日期 2005.10.06
申请人 JANSSEN PHARMACEUTICA, N.V. 发明人 HUANG SHENLIN;LIN RONGHUI;CONNOLLY PETER J.;EMANUEL STUART L.;MIDDLETON STEVEN A.;GRUNINGER ROBERT H.;WETTER STEVEN K.
分类号 A61K31/4196;A61K31/496;A61K33/42;C07D249/14;C07D257/04;C07F9/572;C07F9/6509;C07F9/6515;C07F9/6518 主分类号 A61K31/4196
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