发明名称 PHARMACEUTICAL COMPOSITION COMPRISING IMIDAZOLE CARBONYL COMPOUND
摘要 PROBLEM TO BE SOLVED: To find out that a compound represented by general formula (1), a pharmacologically acceptable salt thereof, and a prodrug thereof have desirable properties as a result of a search for compounds having physical properties of weak cytotoxicity, and high solubility in water, the action to inhibit both of a GyrB subunit of DNA gyrase and a ParE subunit of topoisomerase IV, and sufficient antibacterial activity in order to create an antibiotic having a new mechanism of action. SOLUTION: There is provided a pharmaceutical composition comprising the compound represented by the general formula (1), pharmacologically acceptable salt thereof, and prodrug thereof as an active ingredient (in particular, a composition for preventing or treating infectious diseases). COPYRIGHT: (C)2011,JPO&INPIT
申请公布号 JP2011026305(A) 申请公布日期 2011.02.10
申请号 JP20100142870 申请日期 2010.06.23
申请人 DAIICHI SANKYO CO LTD 发明人 SONEDA GO;TAKESHITA YUTAKA;KAMIKOJIMA KEIKO;YAMAMOTO HIROKO;HOSOKAWA TAKASHI;KONOSU TOSHIYUKI;MASUDA NOBUHISA;UCHIDA TAKUYA;ACHIHA KAZUNARI;KUROYANAGI JUNICHI;FUJISAWA TETSUNORI;YOKOMIZO AKI;NOGUCHI TETSUJI
分类号 A61K31/454;A61K31/407;A61K31/4164;A61K31/4178;A61K31/422;A61K31/427;A61K31/428;A61K31/429;A61K31/4545;A61K31/4709;A61K31/496;A61K31/506;A61K31/538;A61P31/04;A61P43/00 主分类号 A61K31/454
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