发明名称 SF5 DERIVATIVES AS PAR1 INHIBITORS, PRODUCTION THEREOF, AND USE AS MEDICAMENTS
摘要 The invention relates to novel compounds of formula I where R1, R2, R3, R4, R5, R9, Ar, Q1, Q2 and Q3 are each as defined below. The compounds of the formula I have antithrombotic activity and inhibit especially protease-activated receptor 1 (PAR1). The invention further relates to a process for preparing the compound of the formula I and to the use thereof as a medicament.
申请公布号 US2011034461(A1) 申请公布日期 2011.02.10
申请号 US20100851229 申请日期 2010.08.05
申请人 SANOFI-AVENTIS 发明人 HEINELT UWE;WEHNER VOLKMAR;HERRMANN MATTHIAS;SCHOENAFINGER KARL;STEINHAGEN HENNING
分类号 A61K31/5377;A61K31/4035;A61P3/04;A61P7/02;A61P9/06;A61P9/10;A61P29/00;A61P35/00;C07C303/40;C07C381/00;C07D207/06;C07D207/404;C07D209/44;C07D295/112;C07D403/10;C07D413/10 主分类号 A61K31/5377
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