发明名称 AGENT EXHIBITING ANTIPSYCHOTIC ACTIVITY
摘要 FIELD: medicine, pharmaceutics. ^ SUBSTANCE: invention refers to pharmacology and medicine. An agent represents peptide of general formula A-Pro-Tyr-B-X (I) where Pro can represent DPro, A is chosen from Ala, Gly, IIe, Leu, Met, Phe, Ser, Thr, Trp, Tyr, Val; B is chosen from Ala, Arg, Cly, IIe, Leu, Lys, Met, Phe, Pro, Ser, Thr, Trp, Tyr, Val; X-OH; -OCH3; -NH2; -Cly-Pro, and is described as perspective for producing new drugs able to reduce positive and negative symptomatology of schizophrenia and other psychoses. ^ EFFECT: offered is the agent exhibiting antipsychotic activity. ^ 4 dwg, 9 tbl, 15 ex
申请公布号 RU2411248(C2) 申请公布日期 2011.02.10
申请号 RU20080144795 申请日期 2008.11.13
申请人 UCHREZHDENIE ROSSIJSKOJ AKADEMII NAUK INSTITUT MOLEKULJARNOJ GENETIKI RAN (IMG RAN);GOSUDARSTVENNOE UCHREZHDENIE NAUCHNO-ISSLEDOVATEL'SKIJ INSTITUT FARMAKOLOGII IM. V.V. ZAKUSOVA ROSSIJSKOJ AKADEMII MEDITSINSKIKH NAUK (GU NII FARMAKOLOGII IM. V.V. ZAKUSOVA RAMN) 发明人 ANDREEVA LJUDMILA ALEKSANDROVNA;MJASOEDOV NIKOLAJ FEDOROVICH;ZOZULJA ANDREJ ALEKSANDROVICH;KOST NATALIJA VSEVOLODOVNA;MESHAVKIN VIKTOR KONSTANTINOVICH;VORONINA TAT'JANA ALEKSANDROVNA;GARIBOVA TAISIJA LEONOVNA;SEREDENIN SERGEJ BORISOVICH
分类号 A61K38/07;A61K38/08;A61P25/18;C07K5/10;C07K7/06 主分类号 A61K38/07
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