发明名称 |
PROCESS FOR OBTAINING 3,3-DIPHENYLPROPYLAMINES |
摘要 |
<p>The invention relates to a process for obtaining 3,3- diphenylpropylamines of general formula (I), particularly Fesoterodine, as well as their enantiomers, solvates and salts, comprising a chemoselective reduction of the acid group against the ester group in compounds of general formula (V), wherein R1 is C1-C8 alkyl; and R3 and R4, independently of one another, represent H or C1-C8 alkyl, or together form a ring of 3 to 7 members with the nitrogen to which they are bound. The invention also relates to the compounds of formula (V), as well as their enantiomers, solvates and salts.</p> |
申请公布号 |
WO2011012584(A1) |
申请公布日期 |
2011.02.03 |
申请号 |
WO2010EP60817 |
申请日期 |
2010.07.26 |
申请人 |
RAGACTIVES, S.L.U.;LORENTE BONDE-LARSEN, ANTONIO;MARTIN PASCUAL, PABLO;LADERAS MUNOZ, MARIO;GUTIERREZ FUENTES, LUIS GERARDO |
发明人 |
LORENTE BONDE-LARSEN, ANTONIO;MARTIN PASCUAL, PABLO;LADERAS MUNOZ, MARIO;GUTIERREZ FUENTES, LUIS GERARDO |
分类号 |
C07C213/08;C07C219/28 |
主分类号 |
C07C213/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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