摘要 |
DISCLOSED ARE COMPOUNDS AND DERIVATIVES THEREOF, THEIR SYNTHESIS, AND THEIR USE AS RHO-KINASE INHIBITORS. THESE COMPOUNDS OF THE PRESENT INVENTION ARE USEFUL FOR INHIBITING TUMOR GROWTH, TREATING ERECTILE DYSFUNCTION, AND TREATING OTHER INDICATIONS MEDIATED BY RHO-KINASE, E.G., CORONARY HEART DISEASE.
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