发明名称 |
AMINE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONIST ACTIVITY |
摘要 |
Disclosed is an amine derivative of formula (I) where the variable X contains a cyclic group (such as an optionally substituted cycloalkylene) and the other variables are as disclosed in the description. The compounds are useful as NPY Y5 receptor antagonists. Also disclosed is a pharmaceutical composition containing a compound of formula (I) and intermediate compounds used in the preparation of compounds of formula (I). Further disclosed is the use of the compounds in the preparation of a medicament for the treatment of obesity or suppressing food intake.
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申请公布号 |
NZ572381(A) |
申请公布日期 |
2011.01.28 |
申请号 |
NZ20070572381 |
申请日期 |
2007.04.25 |
申请人 |
SHIONOGI & CO., LTD. |
发明人 |
KOUYAMA, NAOKI;OKUNO, TAKAYUKI;SAKAGAMI, MASAHIRO |
分类号 |
C07C311/05;A61K31/18;A61K31/381;A61K31/40;A61K31/415;A61K31/4164;A61K31/4184;A61K31/42;A61P3/04;A61P9/04;A61P15/00;A61P25/08;A61P43/00;C07C311/07;C07C317/36;C07D207/325;C07D211/14;C07D213/38;C07D215/38;C07D217/04;C07D219/10;C07D231/38;C07D233/61;C07D235/30;C07D237/20;C07D239/42;C07D241/20;C07D261/14;C07D263/58;C07D265/30;C07D267/14;C07D275/02;C07D277/28;C07D295/12;C07D333/36;C07D403/04;C07D409/04;C07D413/04;C07D417/12;C07D498/04;C07D513/04 |
主分类号 |
C07C311/05 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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