GAMMA-AMINO-BUTYRIC ACID DERIVATIVES AS GABAB RECEPTOR LIGANDS
摘要
Gamma-amino-butyric acid derivatives of formula (I) that are GABAB receptor ligands, pharmaceutical compositions comprising such derivatives, and methods of using such derivatives and pharmaceutical compositions thereof for treating diseases are disclosed. R5 is chosen from -COOH, -SOOH, and -P(O)(OH)R8 wherein R8 is chosen from hydrogen and C1-4 alkyl.
申请公布号
WO2010120370(A3)
申请公布日期
2011.01.20
申请号
WO2010US01128
申请日期
2010.04.16
申请人
XENOPORT, INC.;XU, FENG;GALLOP, MARK A.;PENG, GE;PHAN, THU;DILIP, USHA;WUSTROW, DAVID J.
发明人
XU, FENG;GALLOP, MARK A.;PENG, GE;PHAN, THU;DILIP, USHA;WUSTROW, DAVID J.