发明名称 AZABICYCLO COMPOUND AND SALT THEREOF
摘要 <p>Disclosed is a novel azabicyclo compound which has both HSP90 inhibitory activity and cell proliferation inhibitory effect. Specifically disclosed is a compound represented by general formula (I) or a salt thereof. (In the formula, X1 represents CH or N; one of X2, X3 and X4 represents N, and the others respectively represent CH; one or two of Y1, Y2, Y3 and Y4 respectively represent C-R4, and the others may be the same or different and respectively represent CH or N; R1 represents an optionally substituted monocyclic or bicyclic unsaturated heterocyclic group that has 1-4 heteroatoms selected from among N, S and O; R2 represents an alkyl group having 1-6 carbon atoms, or the like; and R3 and R4 respectively represent -CO-R5 or the like.)</p>
申请公布号 CA2767556(A1) 申请公布日期 2011.01.13
申请号 CA20102767556 申请日期 2010.07.09
申请人 TAIHO PHARMACEUTICAL CO., LTD. 发明人 KITADE, MAKOTO;OHKUBO, SHUICHI;YOSHIMURA, CHIHOKO;YAMASHITA, SATOSHI;OSHIUMI, HIROMI;UNO, TAKAO;KAWAI, YUICHI
分类号 C07D471/04;A61K31/437;A61K31/444;A61K31/4709;A61K31/5377;A61P35/00;A61P35/02;A61P43/00;C07D519/00 主分类号 C07D471/04
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