发明名称 NOVEL 1,2,3,4-TETRAHYDRO-PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE DERIVATIVES, PREPARATION THEREOF, AND PHARMACEUTICAL USE THEREOF
摘要 The invention relates to the novel materials of formula (I), where: R1 is an optionally substituted L-aryl or –L-heteroaryl, such that L is a single bond, alkyl, CO, or CO-alk, or L'-X, with L' being an alkyl and X being O or S; R2 is H or alkyl; R3 is an alkyl optionally substituted by Hal; and R4 is Hou Hal, wherein said materials are in any isomeric form and the salts thereof, to be used as drugs.
申请公布号 WO2011001113(A2) 申请公布日期 2011.01.06
申请号 WO2010FR51374 申请日期 2010.07.01
申请人 SANOFI-AVENTIS;BACQUE, ERIC;BROLLO, MAURICE;CLAUSS, ANNIE;EL AHMAD, YOUSSEF;FILOCHE-ROMME, BRUNO;HALLEY, FRANK;KARLSSON, KARL ANDREAS;MARCINIAK, GILBERT;RONAN, BAPTISTE;SCHIO, LAURENT;VIVET, BERTRAND;VIVIANI, FABRICE;ZIMMERMANN, ANDRE 发明人 BACQUE, ERIC;BROLLO, MAURICE;CLAUSS, ANNIE;EL AHMAD, YOUSSEF;FILOCHE-ROMME, BRUNO;HALLEY, FRANK;KARLSSON, KARL ANDREAS;MARCINIAK, GILBERT;RONAN, BAPTISTE;SCHIO, LAURENT;VIVET, BERTRAND;VIVIANI, FABRICE;ZIMMERMANN, ANDRE
分类号 C07D487/04;A61K31/519;A61P35/00;C07D239/04;C07D239/06;C07D239/36;C07D239/42;C07D239/47 主分类号 C07D487/04
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