发明名称 |
TRANS-4-[[(5S)-5-[[[3,5-BIS(TRIFLUOROMETHYL)PHENYL]METHYL] (2-METHYL-2H-TETRAZOL-5-YL)AMINO]-2,3,4,5-TETRAHYDRO-7,9-DIMETHYL-1H-1-BENZAZEPIN-1-YL]METHYL]-CYCLOHEXANECARBOXYLIC ACID |
摘要 |
<p>Abstract Compounds of a formula entitled, trans-4-[[(5S)-5-[[[3,5-bis(trifluoromethyl)phenyl]methyl] (2-methyl-2H-tetrazol- 5-yl)amino]-2,3,4,5-tetrahydro-7,9-dimethyl-1H-1-benzazepin-1-yl]methyl]- cyclohexanecarboxylic acid, as a free acid or a pharmaceutically acceptable salt thereof, hydrate, and hydrate in crystalline form; pharmaceutical formulations; and methods of use are disclosed.</p> |
申请公布号 |
WO2011002696(A1) |
申请公布日期 |
2011.01.06 |
申请号 |
WO2010US40125 |
申请日期 |
2010.06.28 |
申请人 |
ELI LILLY AND COMPANY;CHEN, XINCHAO;FRANK, SCOTT, ALAN;REMICK, DAVID, MICHAEL;PEDERSEN, STEVEN, WAYNE |
发明人 |
CHEN, XINCHAO;FRANK, SCOTT, ALAN;REMICK, DAVID, MICHAEL;PEDERSEN, STEVEN, WAYNE |
分类号 |
C07D403/12;A61K31/55;A61P9/10 |
主分类号 |
C07D403/12 |
代理机构 |
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