发明名称 CARBOSTYRIL DERIVATIVES FOR ACCELERATING SALIVATION
摘要 NOVEL PHARMACEUTICAL COMPOSITION FOR ACCELERATING SALIVATION AND FOR PROPHYLAXIS AND/OR TREATMENT OF XEROSTOMIA, WHICH COMPRISES AS AN ACTIVE INGREDIENT A CARBOSTYRIL COMPOUND OF THE FORMULA (1): WHEREIN R IS A HALOGEN ATOM, AND THE SUBSTITUTION POSITION OF THE SUBSTITUENT ON SAID CARBOSTYRIL NUCLEUS IS THE 3- OR 4-POSITION, AND THE BOND BETWEEN THE 3- AND 4- POSITIONS OF THE CARBOSTYRIL NUCLEUS IS EITHER A SINGLE BOND OR A DOUBLE BOND, OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF. THE PHARMACEUTICAL COMPOSITION OF THE PRESENT INVENTION EXHIBITS AN ACCELERATING ACTIVITY OF SALIVATION, AND IS USEFUL IN THE PROPHYLAXIS OR TREATMENT OF XEROSTOMIA OR HYPOSALIVATION.
申请公布号 MY142739(A) 申请公布日期 2010.12.31
申请号 MYPI20042986 申请日期 2004.07.24
申请人 OTSUKA PHARMACEUTICAL CO., LTD.;ST. MARIANNA UNIVERSITY SCHOOL OF MEDICINE 发明人 HISASHI NAGAMOTO;MASAYUKI KOHASHI;HIROSHI OKA
分类号 A61P1/00;A61K31/4704 主分类号 A61P1/00
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