发明名称 |
FUSED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF NUCLEAR HORMONE RECEPTOR FUNCTION |
摘要 |
Disclosed are fused heterocyclic compounds of Formula (I) or pharmaceutically-acceptable salts or stereoisomers thereof. Also disclosed are methods of using such compounds in the treatment of at least one androgen receptor-associated condition, such as, for example, cancer, and pharmaceutical compositions comprising such compounds.
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申请公布号 |
US2010331324(A1) |
申请公布日期 |
2010.12.30 |
申请号 |
US20080666423 |
申请日期 |
2008.06.26 |
申请人 |
BRISTOL-MYERS SQIOBB COMPANY |
发明人 |
NORRIS DEREK J.;GAVAI ASHVINIKUMAR V.;BALOG JAMES AARON;AUSTIN JOEL F.;SHAN WEIFANG;ZHAO YUFEN;NATION ANDREW JAMES;HAN WEN-CHING |
分类号 |
A61K31/5377;A61K31/4035;A61K31/4178;A61K31/4439;A61K31/4709;A61K31/506;A61P17/10;A61P35/00;C07D401/04;C07D401/14;C07D403/14;C07D413/14;C07D491/18 |
主分类号 |
A61K31/5377 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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