发明名称 CRYSTALLINE FORMS OF (3R, 3AS, 6AR) - HEXAHYDROFURO [2,3-B] FURAN-3-YL (1S,2R) - (1-{4-[ (DIETHOXYPHOSPHORYL) METHOXY] PHENY1}-3-HYDROXY-4- [4-METHOXY-N- (2-METHYLPROPYL) BENZENESUL - FONAMIDO] BUTAN-2-YL) CARBAMATE
摘要 The present inventions provides crystaliine forms of (3R,3aS,6aR)- hexahydrofuro[2,3-b]furan-3-yl (1 S,2R)-(1 -{4- [(diethoxyphosphoryl)methoxy]phenyl}-3-hydroxy-4-[4-methoxy-?/-(2- methylpropy[)benzenesulfonamido]butan-2-yl)carbamate, methods of preparing the crystalline forms, pharmaceutical compositions containing the crystalline forms, and therapeutic uses thereof.
申请公布号 WO2010151476(A2) 申请公布日期 2010.12.29
申请号 WO2010US38989 申请日期 2010.06.17
申请人 GILEAD SCIENCES, INC.;CARRA, ERNEST, ANTHONY;CHIU, ANNA;JERNELIUS, JESPER, ALEXIS;WANG, FANG 发明人 CARRA, ERNEST, ANTHONY;CHIU, ANNA;JERNELIUS, JESPER, ALEXIS;WANG, FANG
分类号 C07F9/6561 主分类号 C07F9/6561
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