发明名称 |
CRYSTALLINE FORMS OF (3R, 3AS, 6AR) - HEXAHYDROFURO [2,3-B] FURAN-3-YL (1S,2R) - (1-{4-[ (DIETHOXYPHOSPHORYL) METHOXY] PHENY1}-3-HYDROXY-4- [4-METHOXY-N- (2-METHYLPROPYL) BENZENESUL - FONAMIDO] BUTAN-2-YL) CARBAMATE |
摘要 |
The present inventions provides crystaliine forms of (3R,3aS,6aR)- hexahydrofuro[2,3-b]furan-3-yl (1 S,2R)-(1 -{4- [(diethoxyphosphoryl)methoxy]phenyl}-3-hydroxy-4-[4-methoxy-?/-(2- methylpropy[)benzenesulfonamido]butan-2-yl)carbamate, methods of preparing the crystalline forms, pharmaceutical compositions containing the crystalline forms, and therapeutic uses thereof. |
申请公布号 |
WO2010151476(A2) |
申请公布日期 |
2010.12.29 |
申请号 |
WO2010US38989 |
申请日期 |
2010.06.17 |
申请人 |
GILEAD SCIENCES, INC.;CARRA, ERNEST, ANTHONY;CHIU, ANNA;JERNELIUS, JESPER, ALEXIS;WANG, FANG |
发明人 |
CARRA, ERNEST, ANTHONY;CHIU, ANNA;JERNELIUS, JESPER, ALEXIS;WANG, FANG |
分类号 |
C07F9/6561 |
主分类号 |
C07F9/6561 |
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