发明名称 FUSED OXAZOLE AND THIAZOLE DERIVATIVES AS TRPMS MODULATORS
摘要 The present invention provides fused oxazole and thiazole derivatives as TRPM8 (Transient Receptor Potential subfamily M, member 8) modulators. In particular, compounds described herein are useful for treating diseases, disorders, conditions modulated by TRPM8. Also provided herein are processes for preparing compounds described herein, intermediates used in their synthesis, pharmaceutical compositions thereof, and methods for treating or preventing diseases, conditions and/or disorders modulated by TRPM8.
申请公布号 WO2010010435(A3) 申请公布日期 2010.12.23
申请号 WO2009IB06237 申请日期 2009.07.15
申请人 GLENMARK PHARMACEUTICAL S.A.;IRLAPATI, NAGOSWARA, RAO;THOMAS, ABRAHAM;KURHE, DEEPAK, KANTILAL;SHELKE, SANDEEP, YADUNATH;KHAIRATKAR, JOSHI, NEELIMA;VISWANADHA, SRIKANT;MUKHOPADHYAY, INDRANIL 发明人 IRLAPATI, NAGOSWARA, RAO;THOMAS, ABRAHAM;KURHE, DEEPAK, KANTILAL;SHELKE, SANDEEP, YADUNATH;KHAIRATKAR, JOSHI, NEELIMA;VISWANADHA, SRIKANT;MUKHOPADHYAY, INDRANIL
分类号 C07D263/58;C07D277/82;C07D498/04;C07D513/04 主分类号 C07D263/58
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