发明名称 CARBONATE PRODRUGS AND METHODS OF USING THE SAME.
摘要 The present invention provides carbonate prodrugs which comprise a carbonic phosphoric anhydride prodrug moiety attached to the hydroxyl or carboxyl group of a parent drug moiety. The prodrugs may provide improved physicochemical properties over the parent drug. Also provided are methods of treating a disease or condition that is responsive to the parent drug using the carbonate prodrugs, as well as kits and unit dosages.
申请公布号 MX2010012649(A) 申请公布日期 2010.12.21
申请号 MX20100012649 申请日期 2009.05.20
申请人 NEUROGESX, INC. 发明人 KEITH R. BLEY;NAWEED MUHAMMAD
分类号 A01N57/00 主分类号 A01N57/00
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