发明名称 PREPARATION OF 6-ALPHA-AMINO N-SUBSTITUTED MORPHINANS BY CATALYTIC HYDROGEN TRANSFER
摘要 The present invention provides processes for the stereoselective synthesis of 6-alpha-amino N-substituted morphinans. In particular, the invention provides processes for the reductive amination of 6-keto N-substituted morphinans by catalytic hydrogen transfer.
申请公布号 CA2764915(A1) 申请公布日期 2010.12.16
申请号 CA20102764915 申请日期 2010.06.10
申请人 MALLINCKRODT LLC 发明人 GROTE, CHRISTOPHER W.;CANTRELL, GARY L.;MCCLURG, JOSEPH P.;THOMASSON, CATHERINE E.;MOSER, FRANK W.
分类号 C07D489/00 主分类号 C07D489/00
代理机构 代理人
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