发明名称 |
SALT OF ABT-263 AND SOLID-STATE FORMS THEREOF |
摘要 |
ABT-263 bis-HCl and crystalline polymorphs thereof are suitable active pharmaceutical ingredients for pharmaceutical compositions useful in treatment of a disease characterized by overexpression of one or more anti-apoptotic Bcl-2 family proteins, for example cancer.
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申请公布号 |
US2010305125(A1) |
申请公布日期 |
2010.12.02 |
申请号 |
US20100770345 |
申请日期 |
2010.04.29 |
申请人 |
BORCHARDT THOMAS;BRACKEMEYER PAUL;CATRON NATHANIEL;HENRY RODGER;LOU XIAOCHUN;RAVN MATTHEW;ZHANG GEOFF G Z;ZHOU DELIANG |
发明人 |
BORCHARDT THOMAS;BRACKEMEYER PAUL;CATRON NATHANIEL;HENRY RODGER;LOU XIAOCHUN;RAVN MATTHEW;ZHANG GEOFF G.Z.;ZHOU DELIANG |
分类号 |
A61K31/5377;A61P35/00;A61P35/02;C07D413/12 |
主分类号 |
A61K31/5377 |
代理机构 |
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地址 |
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