PROCESSES FOR THE PREPARATION OF SUBSTITUTED TETRAHYDRO BETA-CARBOLINES
摘要
<p>Provided herein are improved processes for the synthesis of substituted tetrahydro beta-carboline derivatives. In particular, provided herein are improved processes useful for the preparation of (S)-4-chlorophenyl 6-chloro- 1 -(4-methoxyphenyl)-3,4-dihydro- 1 H-pyrido [3,4-b]indole-2(9H)-carboxylate. Formula (I)</p>
申请公布号
WO2010138644(A1)
申请公布日期
2010.12.02
申请号
WO2010US36273
申请日期
2010.05.27
申请人
PTC THERAPEUTICS, INC.;HWANG, PETER, SEONGWOO;MOON, YOUNG-CHOON;ARASU, TAMIL;QI, HONGYAN;ALMSTEAD, NEIL
发明人
HWANG, PETER, SEONGWOO;MOON, YOUNG-CHOON;ARASU, TAMIL;QI, HONGYAN;ALMSTEAD, NEIL