发明名称 PROCESS FOR PREPARATION OF 5-SUBSTITUTED TETRAZOLES
摘要 The present invention is a process for preparing sterically hindered 5-substituted tetrazole, which comprises of reacting a nitrile with an organotin halide and an azide in presence of a phase transfer catalyst, in an organic solvent and a co- solvent at reflux temperature for 4 to 20 h.
申请公布号 WO2010133909(A2) 申请公布日期 2010.11.25
申请号 WO2009IB05660 申请日期 2009.05.20
申请人 SMS PHARMACEUTICALS LIMITED;POTLURI, RAMESH, BABU;DEHURY, SANJAY, KUMAR;VENKATA SUBHRAMANIAN, HARIHARA KRISHNAN 发明人 POTLURI, RAMESH, BABU;DEHURY, SANJAY, KUMAR;VENKATA SUBHRAMANIAN, HARIHARA KRISHNAN
分类号 C07D257/04 主分类号 C07D257/04
代理机构 代理人
主权项
地址