发明名称 |
5-MEMBERED HETEROCYCLIC COMPOUND CYCLOPENTA[C]PYRROLYLALKYLCARBAMATE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF |
摘要 |
<p>The invention relates to compounds of the general formula (I) where: R2 is a hydrogen or fluorine atom or a hydroxyl, cyano, trifluoromethyl, C1-6-alkyl, C1-6-alkoxy, or NR8R9 group; m and p have a value of 1; n and o have the same value which is 0 or 1; A is a covalent bond or a C1-8-alkylene group; R1 is an optionally substituted aryl or heteroaryl group; R3 is a hydrogen or fluorine atom or a C1-6-alkyl group or a trifluoromethyl group; R4 is an optionally substituted 5-membered heterocyclic compound; wherein the compounds can be in the state of a base or an acid addition salt. The present invention can be used in therapeutics.</p> |
申请公布号 |
WO2010130943(A1) |
申请公布日期 |
2010.11.18 |
申请号 |
WO2010FR50912 |
申请日期 |
2010.05.11 |
申请人 |
SANOFI-AVENTIS;ABOUABDELLAH, AHMED;FAYOL, AUDE;LOCHEAD, ALISTAIR;SAADY, MOURAD;VACHE, JULIEN;YAICHE, PHILIPPE |
发明人 |
ABOUABDELLAH, AHMED;FAYOL, AUDE;LOCHEAD, ALISTAIR;SAADY, MOURAD;VACHE, JULIEN;YAICHE, PHILIPPE |
分类号 |
C07D231/12;A61K31/439;A61P25/00;A61P29/00;C07D261/10;C07D277/22;C07D401/14;C07D413/14 |
主分类号 |
C07D231/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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