发明名称 |
Heterocyclic Janus kinase 3 inhibitors |
摘要 |
The invention relates to compound of the formula (I) or its salt, wherein -R 1 , -R 2 , -R 3 , -R 4 , -R 5 , -M-, -X- and -Y= are as defined in the description, their use of as medicament, the process for their preparation and use for the treatment of JAK3 mediated diseases.
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申请公布号 |
EP2251341(A1) |
申请公布日期 |
2010.11.17 |
申请号 |
EP20100174035 |
申请日期 |
2006.07.13 |
申请人 |
ASTELLAS PHARMA INC. |
发明人 |
INOUE, TAKAYUKI;TOJO, TAKASHI;MORITA, MASATAKA;NAKAJIMA, YUTAKA;HATANAKA, KEIKO;SHIRAKAMI, SHOHEI;SASAKI, HIROSHI;TANAKA, AKIRA;TAKAHASHI, FUMIE;MUKOYOSHI, KOICHIRO;HIGASHI, YASUYUKI;OKIMOTO, AKIRA;HONDO, TAKESHI;SAWADA, HITOSHI |
分类号 |
C07D471/04;A61K31/437;A61P11/06;A61P17/00;A61P25/28;A61P35/00;A61P35/02;A61P37/06;C07D471/14;C07D498/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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