发明名称 PROCESS FOR THE MANUFACTURING OF THE COMPOUND 2-HYDROXY-3-[5-(MORPHOLIN-4-YLMETHYL)PYRIDIN-2-YL]1H-INDOLE-5-CARBONITRILE 701
摘要 The present invention relates to a new process for the manufacture of the compound 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1H-indole-5-carbonitrile as a free base and pharmaceutically acceptable salts thereof, particularly the 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1H-indole-5-carbonitrile citrate, and to new intermediates prepared in said process suitable for large scale manufacturing of said compound.
申请公布号 US2010286392(A1) 申请公布日期 2010.11.11
申请号 US20080596020 申请日期 2008.04.17
申请人 DELISSER VERN;HEDBERG MARTIN;JANSSON ANNETTE;RADEVIK ANDREAS;RYBERG PER;THIERING SWANTJE 发明人 DELISSER VERN;HEDBERG MARTIN;JANSSON ANNETTE;RADEVIK ANDREAS;RYBERG PER;THIERING SWANTJE
分类号 C07D413/06;C07D413/14 主分类号 C07D413/06
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