发明名称 PREPARATION METHOD OF STATIN COMPOUND AND BENZOTHIAZOLYL SULFONE COMPOUND USED THEREIN
摘要 The inventive method comprising subjecting a novel benzothiazolyl sulfone compound to a reaction with an aldehyde to obtain a vinyl intermediate and removing the hydroxy and carboxy protective groups of the vinyl intermediate is simple and efficient in preparing a statin compound or a salt thereof which is useful for treating hyperlipemia.
申请公布号 WO2010077062(A3) 申请公布日期 2010.11.04
申请号 WO2009KR07881 申请日期 2009.12.29
申请人 HANMI PHARM. CO., LTD.;KIM, HEE SEOCK;KIM, WON JEOUNG;KIM, HEE CHEOL;SIM, JAE YI;CHO, SEONG MI;BYUN, EUN YOUNG;JEON, JI YOUNG;LEE, YOON JU;SUH, KWEE HYUN;LEE, GWAN SUN 发明人 KIM, HEE SEOCK;KIM, WON JEOUNG;KIM, HEE CHEOL;SIM, JAE YI;CHO, SEONG MI;BYUN, EUN YOUNG;JEON, JI YOUNG;LEE, YOON JU;SUH, KWEE HYUN;LEE, GWAN SUN
分类号 C07D239/18;C07D215/02 主分类号 C07D239/18
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