发明名称 |
STABILIZED LIPID FORMULATION OF APOPTOSIS PROMOTER |
摘要 |
An orally deliverable pharmaceutical composition comprises a Bcl-2 family protein inhibitory compound, e.g., ABT-263, a heavier-chalcogen antioxidant and a substantially non-aqueous lipid carrier, wherein said compound and said antioxidant are in solution in the carrier. The composition is suitable for oral administration to a subject in need thereof for treatment of a disease characterized by overexpression of one or more anti-apoptotic Bcl-2 family proteins, for example cancer.
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申请公布号 |
US2010278905(A1) |
申请公布日期 |
2010.11.04 |
申请号 |
US20100770174 |
申请日期 |
2010.04.29 |
申请人 |
CATRON NATHANIEL;FICKES MICHAEL G;FISCHER CRISTINA M;HAIGHT ANTHONY R;HEEMSTRA KATHERINE;SANZGIRI YESHWANT D;SCHMITT ERIC A;TONG PING;ZHANG GEOFF G Z;ZHOU DELIANG |
发明人 |
CATRON NATHANIEL;FICKES MICHAEL G.;FISCHER CRISTINA M.;HAIGHT ANTHONY R.;HEEMSTRA KATHERINE;SANZGIRI YESHWANT D.;SCHMITT ERIC A.;TONG PING;ZHANG GEOFF G. Z.;ZHOU DELIANG |
分类号 |
A61K31/5377;A61K9/127;A61K9/66;A61P35/00;A61P35/02 |
主分类号 |
A61K31/5377 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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