发明名称 |
PROCESS FOR MAKING (R) -3-(2,3-DIHYDROXYPROPYL)-6-FLUORO-5-(2-FLOURO-4-IODOPHENYLAMINO)-8-METHYLPYRIDO[2,3-d]PYRIMIDINE-4,7(3H,8H)-DIONE AND INTERMEDIATES THEREOF |
摘要 |
The present invention relates generally to processes of making (R)-3-(2,3-Dihydroxypropyl)-6-fluoro-5-(2-fluoro-4-iodophenylamino)-8-methylpyrido[2,3-d]pyrimidine-4,7(3H,8H)-dione, intermediates thereof, and a process for making a particular polymorph of (R)-3-(2,3-Dihydroxypropyl)-6-fluoro-5-(2-fluoro-4-iodophenylamino)-8-methylpyrido[2,3-d]pyrimidine-4,7(3H,8H)-dione. |
申请公布号 |
WO2010059503(A3) |
申请公布日期 |
2010.11.04 |
申请号 |
WO2009US64218 |
申请日期 |
2009.11.12 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED;PROVENCAL, DAVID, PAUL;MILLER, TODD;ZHAO, YUXIN;SALSBURY, JONATHON, S. |
发明人 |
PROVENCAL, DAVID, PAUL;MILLER, TODD;ZHAO, YUXIN;SALSBURY, JONATHON, S. |
分类号 |
C07D213/82;C07C255/23;C07D213/85;C07D471/04 |
主分类号 |
C07D213/82 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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