发明名称 |
PROCESS FOR THE PREPARATION OF BENZO-FUSED HETEROARYL SULFAMATES AND CRYSTALLINE FORM OF N- ( ( (2S) -6-CHLORO-2,3-DIHYDRO-L,4-BE NZODIOXIN-2-YL) METHYL-SULFAMIDE. |
摘要 |
<p>The present invention is directed to a process for the preparation of benzo-fused heteroaryl sulfamates, useful for the treatment of epilepsy and related disorders according to formula (IA) and to a crystalline compound of formula (I-S). Process for the preparation of a compound of formula (IA).</p> |
申请公布号 |
MX2010010595(A) |
申请公布日期 |
2010.10.25 |
申请号 |
MX20100010595 |
申请日期 |
2008.03.26 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
MEHRMAN, STEVEN J.;ABDEL-MAGID, AHMED F. |
分类号 |
C07D311/58;A61K31/357;A61P25/08;C07D317/58;C07D319/20;C07D321/08 |
主分类号 |
C07D311/58 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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