发明名称 PROCESS FOR THE PREPARATION OF BENZO-FUSED HETEROARYL SULFAMATES AND CRYSTALLINE FORM OF N- ( ( (2S) -6-CHLORO-2,3-DIHYDRO-L,4-BE NZODIOXIN-2-YL) METHYL-SULFAMIDE.
摘要 <p>The present invention is directed to a process for the preparation of benzo-fused heteroaryl sulfamates, useful for the treatment of epilepsy and related disorders according to formula (IA) and to a crystalline compound of formula (I-S). Process for the preparation of a compound of formula (IA).</p>
申请公布号 MX2010010595(A) 申请公布日期 2010.10.25
申请号 MX20100010595 申请日期 2008.03.26
申请人 JANSSEN PHARMACEUTICA N.V. 发明人 MEHRMAN, STEVEN J.;ABDEL-MAGID, AHMED F.
分类号 C07D311/58;A61K31/357;A61P25/08;C07D317/58;C07D319/20;C07D321/08 主分类号 C07D311/58
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