发明名称 |
ABCG2 INHIBITOR |
摘要 |
The present invention relates to a breast cancer resistance protein (BCRP/ABCG2) inhibitor. The invention provides an acrylonitrile derivative represented by formula (1): (wherein A represents an optionally substituted 3- to 8-membered heterocyclic ring) or a salt thereof.
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申请公布号 |
US2010249089(A1) |
申请公布日期 |
2010.09.30 |
申请号 |
US20080745899 |
申请日期 |
2008.12.02 |
申请人 |
KABUSHIKI KAISHA YAKULT HONSHA |
发明人 |
YAMAZAKI RYUTA;HATANO HIROSHI;YAEGASHI TAKASHI;IGARASHI YOSHIAKI;YOSHIDA OH;SUGIMOTO YOSHIKAZU |
分类号 |
A61K31/4545;A61K31/4535;A61K31/454;A61K31/496;A61K31/5377;A61P35/00;C07D409/14 |
主分类号 |
A61K31/4545 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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