发明名称 ABCG2 INHIBITOR
摘要 The present invention relates to a breast cancer resistance protein (BCRP/ABCG2) inhibitor. The invention provides an acrylonitrile derivative represented by formula (1): (wherein A represents an optionally substituted 3- to 8-membered heterocyclic ring) or a salt thereof.
申请公布号 US2010249089(A1) 申请公布日期 2010.09.30
申请号 US20080745899 申请日期 2008.12.02
申请人 KABUSHIKI KAISHA YAKULT HONSHA 发明人 YAMAZAKI RYUTA;HATANO HIROSHI;YAEGASHI TAKASHI;IGARASHI YOSHIAKI;YOSHIDA OH;SUGIMOTO YOSHIKAZU
分类号 A61K31/4545;A61K31/4535;A61K31/454;A61K31/496;A61K31/5377;A61P35/00;C07D409/14 主分类号 A61K31/4545
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