发明名称 |
LIGANDS FOR TRANSITION-METAL-CATALYZED CROSS-COUPLINGS, AND METHODS OF USE THEREOF |
摘要 |
<p>Ligands for transition metals are disclosed herein, which may be used in various transition-metal-catalyzed carbon-heteroatom and carbon-carbon bond-forming reactions. The disclosed methods provide improvements in many features of the transition-metal-catalyzed reactions, including the range of suitable substrates, number of catalyst turnovers, reaction conditions, and efficiency. For example, improvements have been realized in transition-metal-catalyzed cross-coupling reactions.</p> |
申请公布号 |
EP2231680(A2) |
申请公布日期 |
2010.09.29 |
申请号 |
EP20080860439 |
申请日期 |
2008.12.12 |
申请人 |
MASSACHUSETTS INSTITUTE OF TECHNOLOGY |
发明人 |
BUCHWALD, STEPHEN, L.;FORS, BRETT, P.;SURRY, DAVID, S. |
分类号 |
C07F9/02;C07C209/10;C07C213/00;C07C231/08;C07D213/74;C07D241/20;C07D401/12;C07D403/04;C07F9/50;C07F15/00 |
主分类号 |
C07F9/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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