发明名称 PROCESS FOR PREPARATION OF 4-(3'-CHLORO-4'-FLUOROANILINO)-7-METHOXY-6-(3-MORPHOLINOPROPOXY)QUINAZOLINE
摘要 <P>PROBLEM TO BE SOLVED: To provide a means useful for preparing a pharmacologically effective quinazoline derivative. Ž<P>SOLUTION: Intermediates of compounds of formula II and formula III are useful in a method for preparing a pharmacologically effective quinazoline derivative such as a quinazoline derivative and 4-(3'-chloro-4'-fluoroanilino)-7-methoxy-6-(3-morpholinopropoxy)quinazoline, respectively. Ž<P>COPYRIGHT: (C)2010,JPO&INPIT Ž
申请公布号 JP2010209071(A) 申请公布日期 2010.09.24
申请号 JP20100061976 申请日期 2010.03.18
申请人 ASTRAZENECA AB 发明人 GILDAY JOHN PETER;MOODY DAVID
分类号 C07D413/12;C07D239/88;C07D239/94;C07D265/30;C07D295/092 主分类号 C07D413/12
代理机构 代理人
主权项
地址