发明名称 |
PROCESS FOR PREPARATION OF 4-(3'-CHLORO-4'-FLUOROANILINO)-7-METHOXY-6-(3-MORPHOLINOPROPOXY)QUINAZOLINE |
摘要 |
<P>PROBLEM TO BE SOLVED: To provide a means useful for preparing a pharmacologically effective quinazoline derivative. Ž<P>SOLUTION: Intermediates of compounds of formula II and formula III are useful in a method for preparing a pharmacologically effective quinazoline derivative such as a quinazoline derivative and 4-(3'-chloro-4'-fluoroanilino)-7-methoxy-6-(3-morpholinopropoxy)quinazoline, respectively. Ž<P>COPYRIGHT: (C)2010,JPO&INPIT Ž
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申请公布号 |
JP2010209071(A) |
申请公布日期 |
2010.09.24 |
申请号 |
JP20100061976 |
申请日期 |
2010.03.18 |
申请人 |
ASTRAZENECA AB |
发明人 |
GILDAY JOHN PETER;MOODY DAVID |
分类号 |
C07D413/12;C07D239/88;C07D239/94;C07D265/30;C07D295/092 |
主分类号 |
C07D413/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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