发明名称 GLYCINE TRANSPORTER INHIBITOR
摘要 <p>Provided is a novel compound or a pharmaceutically acceptable salt thereof, which is useful for preventing or treating diseases attributed to glycine uptake inhibitory activity such as schizophrenia, Alzheimer's disease, cognitive impairment, dementia, anxiety disorders (such as generalized anxiety disorders, panic disorders, obsessive-compulsive disorders, social anxiety disorders, post-traumatic stress disorders, specific phobia, and acute stress disorders), depression, drug dependence, convulsion, tremor, and sleep disorders. The compound is represented by formula [I].</p>
申请公布号 WO2010107115(A1) 申请公布日期 2010.09.23
申请号 WO2010JP54831 申请日期 2010.03.19
申请人 TAISHO PHARMACEUTICAL CO., LTD.;YASUHARA, AKITO;YAMAMOTO, SHUJI;OHTA, HIROSHI;SHIRASAKI, YOSHIHISA;SAKAGAMI, KAZUNARI;HAYASHI, MASATO;SHIBATA, TSUYOSHI;SHIMAZAKI, YOUICHI;ARAKI, YUKO;ABE, KUMI;SUN, XIANG-MIN 发明人 YASUHARA, AKITO;YAMAMOTO, SHUJI;OHTA, HIROSHI;SHIRASAKI, YOSHIHISA;SAKAGAMI, KAZUNARI;HAYASHI, MASATO;SHIBATA, TSUYOSHI;SHIMAZAKI, YOUICHI;ARAKI, YUKO;ABE, KUMI;SUN, XIANG-MIN
分类号 C07D405/12;A61K31/4178;A61K31/4196;A61K31/437;A61K31/4439;A61P25/08;A61P25/14;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P43/00;C07D405/14;C07D409/12;C07D471/04 主分类号 C07D405/12
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