发明名称 |
Process for Preparing (S)-(+)-N-Methyl-3-(1-Naphthyloxy)-3-(2-Thienyl-Propylamine by using Optically Active Methylhydroxylaminopropanol Compound as an Intermediate |
摘要 |
<p>The present invention provides a ( S )-methylhydroxylaminopropanol compound as an intermediate for preparation of ( S )-(+)- N -methyl-3-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propylamine. The present invention also provides a process for preparing ( S )-(+)- N -methyl-3-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propylamine with higher yield and low treatment cost, which includes a process for preparing a N -methyl- N -hydroxyl-3-(1-naphthyloxy)-3-(2-thienyl)propylamine compound.</p> |
申请公布号 |
EP2228372(A1) |
申请公布日期 |
2010.09.15 |
申请号 |
EP20100156142 |
申请日期 |
2010.03.10 |
申请人 |
SCI PHARMATECH, INC. |
发明人 |
CHEN, BO-FENG;YEH, JINUN-BAN;WONG, WEICHYUN;LU, FENG-JU |
分类号 |
C07D333/16 |
主分类号 |
C07D333/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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