发明名称 Process for Preparing (S)-(+)-N-Methyl-3-(1-Naphthyloxy)-3-(2-Thienyl-Propylamine by using Optically Active Methylhydroxylaminopropanol Compound as an Intermediate
摘要 <p>The present invention provides a ( S )-methylhydroxylaminopropanol compound as an intermediate for preparation of ( S )-(+)- N -methyl-3-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propylamine. The present invention also provides a process for preparing ( S )-(+)- N -methyl-3-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propylamine with higher yield and low treatment cost, which includes a process for preparing a N -methyl- N -hydroxyl-3-(1-naphthyloxy)-3-(2-thienyl)propylamine compound.</p>
申请公布号 EP2228372(A1) 申请公布日期 2010.09.15
申请号 EP20100156142 申请日期 2010.03.10
申请人 SCI PHARMATECH, INC. 发明人 CHEN, BO-FENG;YEH, JINUN-BAN;WONG, WEICHYUN;LU, FENG-JU
分类号 C07D333/16 主分类号 C07D333/16
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