发明名称 PROCESS FOR PRODUCING PYRROLE COMPOUND
摘要 A process for producing a sulfonylpyrrole compound useful as a medicine, a process for producing an intermediate for use in the process, and a novel intermediate. The process for producing a sulfonylpyrrole compound (VIII) comprises reducing a compound (III), subsequently hydrolyzing the compound to obtain a compound (IV), sulfonylating the compound (IV) to obtain a compound (VI), and aminating the compound (VI) to thereby produce the compound (VIII).
申请公布号 WO2010098351(A1) 申请公布日期 2010.09.02
申请号 WO2010JP52874 申请日期 2010.02.24
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;IKEMOTO, TOMOMI;MIZUFUNE, HIDEYA;NAGATA, TOSHIAKI;SERA, MISAYO;FUKUDA, NAOHIRO;YAMASAKI, TAKESHI 发明人 IKEMOTO, TOMOMI;MIZUFUNE, HIDEYA;NAGATA, TOSHIAKI;SERA, MISAYO;FUKUDA, NAOHIRO;YAMASAKI, TAKESHI
分类号 C07D207/34;C07D207/333;C07D207/36;C07D401/12 主分类号 C07D207/34
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