发明名称 FUSED HETEROCYCLIC RING COMPOUND
摘要 <p>Disclosed is a compound represented by formula (I) or a salt thereof, which has GPR 119 agonist action and excellent medicinal effects useful for prevention/treatment of diabetes, adiposis and the like. In the formula, P represents a substituted 6-membered aromatic ring; Q represents a (substituted) 6-membered aromatic ring; A1 represents CR4aR4b, NR4c, O, S, SO, SO2 (wherein R4a-R4c each represents H or the like); L1 represents a (substituted) C1-5 alkylene; L2 represents a bond, a (substituted) C1-3 alkylene; L3 and L4 each represents a (substituted) C1-3 alkylene; R1 represents H, X, CN, a (substituted) hydrocarbon, a (substituted) heterocyclic ring or a (substituted) OH, or alternatively combines with A1 to form a (substituted) 4- to 8-membered (heterocyclic) ring; R2 represents H, CN or a (substituted) hydrocarbon; and R3a represents -COSRA1 or a (substituted) 5- or 6-membered aromatic ring (wherein RA1 represents a (substituted) hydrocarbon or a (substituted) heterocyclic ring).)</p>
申请公布号 WO2010095663(A1) 申请公布日期 2010.08.26
申请号 WO2010JP52374 申请日期 2010.02.17
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;RIKIMARU, KENTARO;IMOTO, HIROSHI;KAMAURA, MASAHIRO 发明人 RIKIMARU, KENTARO;IMOTO, HIROSHI;KAMAURA, MASAHIRO
分类号 C07D401/14;A61K31/454;A61K31/506;A61K31/519;A61K31/5377;A61K31/55;A61P1/00;A61P1/02;A61P1/04;A61P1/08;A61P1/12;A61P1/16;A61P1/18;A61P3/04;A61P3/06;A61P3/10;A61P7/00;A61P9/00;A61P9/04;A61P9/10;A61P9/12;A61P11/00;A61P13/10;A61P13/12;A61P15/00;A61P17/02;A61P17/06;A61P19/02;A61P19/06;A61P19/10;A61P21/04;A61P25/00;A61P25/02;A61P25/28;A61P27/02;A61P27/12;A61P27/16;A61P29/00;A61P31/00;A61P35/00;A61P35/02;A61P43/00;C07D405/14;C07D413/14;C07D487/04 主分类号 C07D401/14
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